63427-91-8Relevant academic research and scientific papers
Synthesis and Evaluation of a Mitochondria-Targeting Poly(ADP-ribose) Polymerase-1 Inhibitor
Krainz, Tanja,Lamade, Andrew M.,Du, Lina,Maskrey, Taber S.,Calderon, Michael J.,Watkins, Simon C.,Epperly, Michael W.,Greenberger, Joel S.,Baylr, Hülya,Wipf, Peter,Clark, Robert S. B.
, p. 2868 - 2879 (2018/09/25)
The poly(ADP-ribose) polymerase (PARP) family of enzymes plays a crucial role in cellular and molecular processes including DNA damage detection and repair and transcription; indeed, PARP inhibitors are under clinical evaluation as chemotherapeutic adjunc
BENZOXAZOLE CARBOXAMIDE INHIBITORS OF POLY(ADP-RIBOSE)POLYMERASE (PARP)
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Page/Page column 72, (2009/08/16)
A compound having the structure set forth in Formula (I) or Formula (II): wherein the variables Y, R1, R2, R3, and R4 are as defined herein. Provided herein are inhibitors of poly(ADP-ribose)polymerase activity. Also described herein are pharmaceutical compositions that include at least one compound described herein and the use of a compound or pharmaceutical composition described herein to treat diseases, disorders and conditions that are ameliorated by the inhibition of PARP activity.
1H-benzimidazole-4-carboxamides substituted with a quaternary carbon at the 2-position are potent PARP inhibitors
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Page/Page column 14, (2008/06/13)
Compounds of Formula (I) inhibit the PARP enzyme and are useful for treating a disease or a disorder associated with PARP. Also disclosed are pharmaceutical compositions comprising compounds of Formula (I), methods of treatment comprising compounds of For
Preparation, Isolation and X-Ray Crystallographic Structure Determination of a Stable, Crystalline Carbonic Anhydride of an N-Protected α-Amino Acid
Chan, Chat-On,Cooksey, Christopher J.,Crich, David
, p. 777 - 780 (2007/10/02)
The reaction of methyl (2S,3aR,8aS)-2-carboxy-8-phenylsulfonyl-1,2,3,3a,8,8a-hexahydropyrrolo-indole-1-carboxylate and isobutyl chloroformate in tetrahydrofuran at -15 deg C in the presence of trimethylamine results in the formation of the correspo
