661467-30-7Relevant articles and documents
Na+-dependent high affinity binding of [3H]LY515300, a 3,4-dimethyl-4-(3-hydroxyphenyl)piperidine opioid receptor inverse agonist
Statnick, Michael A.,Suter, Todd M.,Gackenheimer, Susan L.,Emmerson, Paul J.,Quimby, Steve J.,Gehlert, Donald R.,Wheeler, William J.,Mitch, Charles H.
, p. 139 - 150 (2003)
Analogues of 3,4-dimethyl-4-(3-hydroxyphenyl)piperidines are high affinity inverse agonists for μ-, δ- and κ-opioid receptors. To characterize inverse agonist binding, we synthesized a high specific activity radioligand from this series, [3H]LY