67413-25-6Relevant articles and documents
COVALENT RAS INHIBITORS AND USES THEREOF
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Page/Page column 175, (2021/06/04)
The disclosure features compounds, or pharmaceutically acceptable salts thereof, alone and in combination with other therapeutic agents, pharmaceutical compositions, and protein conjugates thereof, capable of modulating biological processes including Ras, and their uses in the treatment of cancers.
Genetic encoding of 2-aryl-5-carboxytetrazole-based protein photo-cross-linkers
Tian, Yulin,Lin, Qing
, p. 4449 - 4452 (2018/05/03)
Three γ-heteroatom-substituted N-methylpyrroletetrazole-lysines (mPyTXKs) were synthesized and subsequently incorporated into proteins site-specifically via genetic code expansion. The γ-seleno-substituted derivative, mPyTSeK, showed excellent incorporati
Synthesis of natural and non natural orthogonally protected lanthionines from N-tritylserine and allo-threonine derivatives
Dugave, Christophe,Menez, Andre
, p. 1453 - 1465 (2007/10/03)
The reactivity of electrophiles derived from N-tritylserine, threonine and allothreonine esters toward a selection of nucleophiles was investigated. Best yields from substitution products were obtained with N-trityliodoalanine and soft nucleophiles such a