689290-83-3Relevant articles and documents
4-[6-(2-Aminoethyl)naphthalen-2-yl]benzonitriles are potent histamine H3 receptor antagonists with high CNS penetration
Black, Lawrence A.,Nersesian, Diana L.,Sharma, Padam,Ku, Yi-Yin,Bennani, Youssef L.,Marsh, Kennan C.,Miller, Thomas R.,Esbenshade, Timothy A.,Hancock, Arthur A.,Cowart, Marlon
, p. 1443 - 1446 (2007/10/03)
4-[6-(2-Tertiaryaminoethyl)naphthalen-2-yl]benzonitriles are conformationally constrained histamine H3 receptor antagonists with high potency and selectivity. The analogs were designed around a naphthalene core, with the goal of enhancing lipop