69135-70-2Relevant academic research and scientific papers
Endothelin receptor antagonists: Synthesis and structure-activity relationships of substituted benzothiazine-1,1-dioxides
Berryman,Edmunds,Bunker,Haleen,Bryant,Welch,Doherty
, p. 1447 - 1456 (2007/10/03)
The development of benzothiazine-1,1-dioxide derivatives as a new structural class of potent endothelin receptor antagonists is described. Structure-activity relationships (SAR) revealed that PD164800 (1) is a potent antagonist of the ET(A) receptor subtype. Copyright (C) 1998 Elsevier Science Ltd.
3,3'-Bis-methylene-1,3-benzo-thiazine compounds
-
, (2008/06/13)
3,3'-Bis-Methylene-1,3-benzothiazine compounds are inhibitors of phenylethanolamine N-methyl-transferase.
