70959-58-9Relevant academic research and scientific papers
Discovery of novel CDK inhibitors via scaffold hopping from CAN508
Jing, Liandong,Tang, Yanbo,Xiao, Zhiyan
supporting information, p. 1386 - 1391 (2018/03/21)
Cyclin-dependent kinases (CDKs) are promising drug targets for various human diseases, especially for cancers. Scaffold hopping strategy was applied on CAN508, a known selective CDK9 inhibitor, and a series of pyrazolo[3,4-b]pyridine compounds were synthe
