70963-39-2Relevant articles and documents
Facile synthesis of highly functionalized N-methyl amino acid esters without side-chain protection
White, Kimberly N.,Konopelski, Joseph P.
, p. 4111 - 4112 (2007/10/03)
(Chemical Equation Presented) The facile, two-pot synthesis of N-methyl amino acid esters by way of reductive amination is presented. Side chain protection schemes are not required, the starting materials are all commercially available, and the synthetic
Immonium Ion Based Synthetic Methodology: A Novel Method for the N-Methylation of Dipeptides and Amino Acid Derivatives via Retro Aza Diels-Alder Reactions
Grieco, Paul A.,Bahsas, Ali
, p. 5746 - 5749 (2007/10/02)
A novel method for the N-methylation of amino acid derivatives and dipeptides is detailed that features facile room-temperature retro Diels-Alder reactions of N-substituted 2-azanorbornenes with trapping of the incipient immonium ion with triethylsilane/trifluoroacetic acid.
Tumor-resolving and histolytic medicaments and their use
-
, (2008/06/13)
Dehydrooligopeptides, some of which are known, demonstrate histolytic and tumor-resolving activity and may be used in medicaments causing the lysis of animal tissues and/or tumors in warm-blooded animals.