70998-42-4Relevant articles and documents
Tri- and tetrasubstituted pyridinylimidazoles as covalent inhibitors of c-Jun N-terminal kinase 3
Muth, Felix,El-Gokha, Ahmed,Ansideri, Francesco,Eitel, Michael,D?ring, Eva,Sievers-Engler, Adrian,Lange, Andreas,Boeckler, Frank M.,L?mmerhofer, Michael,Koch, Pierre,Laufer, Stefan A.
, p. 594 - 607 (2017/02/05)
The concept of covalent inhibition of c-Jun N-terminal kinase 3 (JNK3) was successfully transferred to our well validated pyridinylimidazole scaffold varying several structural features in order to deduce crucial structure-activity relationships. Joint ta