754987-62-7Relevant academic research and scientific papers
UNUSUAL SUBSTRATES OF TUBULIN TYROSINE LIGASE
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Page/Page column 90, (2017/12/09)
The present invention provides means and methods for functionalizing a polypeptide of interest at its C-terminus with an amino acid derivative.
A facile transformation of amino acids to functionalized coumarins
Bandyopadhyay, Anupam,Gopi, Hosahudya N.
supporting information; experimental part, p. 8089 - 8095 (2012/01/04)
The synthesis of novel chiral coumarins functionalized with proteinogenic amino acid side chains via N-protected γ-amino-β-keto esters and their incorporation into the cell permeable HIV-1 TAT peptide through the modified solid phase peptide synthesis are
Tin(ii) chloride assisted synthesis of N-protected γ-amino β-keto esters through semipinacol rearrangement
Bandyopadhyay, Anupam,Agrawal, Neha,Mali, Sachitanand M.,Jadhav, Sandip V.,Gopi, Hosahudya N.
experimental part, p. 4855 - 4860 (2010/12/24)
A facile synthetic route for the preparation of N-protected γ-amino β-keto esters from amino aldehydes and ethyl diazoacetate is described. The two component coupling is facilitated by tin(ii) chloride followed by semipinacol rearrangement leading to the product in quantitative yield. The reaction is mild, instantaneous and compatible with Boc-, Fmoc- and Cbz-amino protecting groups.
A method for manufacturing optically active coumaryl amino acid salts and the coumaryl aminoacid salts thus obtained
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Page/Page column 13, (2010/02/13)
The present invention relates to the field of the synthesis of optically active amino acids, mainly for the purpose of manufacturing optically active polypeptides that are useful as labelled detection tools. The manufacturing method involves the preparati
A very short route to enantiomerically pure coumarin-bearing fluorescent amino acids
Brun, Marie-Priscille,Bischoff, Laurent,Garbay, Christiane
, p. 3432 - 3436 (2007/10/03)
No bulkier than a tryptophan or a tyrosine residue are the fluorescent coumaryl amino acids described. These building blocks can be synthesized rapidly with high enantiomeric purity and introduced readily into a peptidic sequence. Their fluorescence prope
