78471-81-5Relevant academic research and scientific papers
Design, synthesis and evaluation of benzoisothiazolones as selective inhibitors of PHOSPHO1
Bravo, Yalda,Teriete, Peter,Dhanya, Raveendra-Panickar,Dahl, Russell,Lee, Pooi San,Kiffer-Moreira, Tina,Ganji, Santhi Reddy,Sergienko, Eduard,Smith, Layton H.,Farquharson, Colin,Millan, Jose Luis,Cosford, Nicholas D.P.
, p. 4308 - 4311 (2014/09/17)
We report the discovery and characterization of a series of benzoisothiazolone inhibitors of PHOSPHO1, a newly identified soluble phosphatase implicated in skeletal mineralization and soft tissue ossification abnormalities. High-throughput screening (HTS)
Phenyliodine(III) bis(trifluoroacetate) mediated synthesis of 2-aryl-1,2-benzisothiazol-3(2H)-ones in ionic liquid
Wang, Huey-Min,Liang, I.-Chian,Hou, Rei-Sheu,Huang, Hsin-Yu,Chen, Ling-Ching
, p. 127 - 130 (2008/02/11)
Treatment of N-aryl-2-(benzylthio)benzamides with phenyliodine(III) bis(trifluoroacetate) containing trifluoroacetic acid resulted in an interrupted Pummerer-type reaction in ionic liquid 1-n-butyl-3-methylimidazolium hexafluorophosphate, [bmim][PF6
An interrupted Pummerer reaction induced by hypervalent iodine(III) reagent: Facile synthesis of 2-aryl-1,2-benzisothiazol-3(2H)-ones
Wang, Huey-Min,Huang, Hsin-Yu,Kang, Iou-Jiun,Chen, Ling-Ching
, p. 1231 - 1235 (2007/10/03)
Treatment of N-aryl-2-(benzylthio)benzamides with phenyliodine(III) bis(trifluoroacetate) containing trifluoroacetic acid resulted in an interrupted Pummerer-type reaction to give 2-aryl-1,2-benzisothiazol-3(2H)-ones rather than the normal Pummerer-type p
