791122-48-0Relevant academic research and scientific papers
NO-sartans: A new class of pharmacodynamic hybrids as cardiovascular drugs
Breschi, Maria C.,Calderone, Vincenzo,Digiacomo, Maria,Martelli, Alma,Martinotti, Enrica,Minutolo, Filippo,Rapposelli, Simona,Balsamo, Aldo
, p. 5597 - 5600 (2004)
The aim of this work was to develop lead pharmacodynamic hybrids, NO-sartans, possessing the characteristics of a typical AT1- antagonist and of a "slow NO donor", by adding NO-donor side chains to losartan. These new compounds, 2a and 2b, disp
