797049-66-2Relevant academic research and scientific papers
N-alkylation of N-arylsulfonyl-α-amino acid methyl esters by trialkyloxonium tetrafluoroborates
De Marco, Rosaria,Di Gioia, Maria Luisa,Liguori, Angelo,Perri, Francesca,Siciliano, Carlo,Spinella, Mariagiovanna
supporting information; experimental part, p. 9708 - 9714 (2012/01/03)
In this work we present the results obtained for the N-alkylation of a series of N-arylsulfonyl-α-amino acid methyl esters bearing different substituents at the 4-position of the sulfonamide aromatic ring. In particular, we compare the reactivity of these
Peptidic aldehydes based on α- and β-amino acids: Synthesis, inhibition of m-Calpain, and anti-cataract properties
Payne, Richard J.,Brown, Karina M.,Coxon, James M.,Morton, James D.,Lee, Hannah Yun-Young,Abell, Andrew D.
, p. 877 - 884 (2007/10/03)
We present a new synthesis of SJA6017 (a potent m-calpain inhibitor) and its adaptation in order to prepare analogues in which the constituent Leu and Val residues are systematically replaced with their corresponding β-amino acids and/or the N-terminal fl
