80517-23-3

Upstream product

• 446-32-2 4-fluoroanthranilic acid 
• 98-59-9 p-toluenesulfonyl chloride 
• 456-22-4 4-Fluorobenzoic acid 
• 1570134-76-7 N-(2-(4,5-dihydrooxazol-2-yl)phenyl)-4-fluorobenzamide 
• 403-43-0 4-fluorobenzoyl chloride 
• 1570135-10-2 N-(2-(4,5-dihydrooxazol-2-yl)phenyl)-4-fluoro-2-(4-methylphenylsulfonamido)benzamide 

Downstream Products

• 1392300-33-2 N-(5-fluoro-2-(hydrazinecarbonyl)phenyl)-4-methylbenzenesulfonamide 

Relevant academic research and scientific papers

INHIBITORS OF OPLOPHORUS LUCIFERASE-DERIVED BIOLUMINESCENT COMPLEXES

Compounds that may selectively inhibit Oplophorus luciferase-derived bioluminescent complexes, e.g., NanoBiT? bioluminescent complex, are disclosed as well as compositions and kits comprising the compounds, and methods of using the compounds. The compounds are of formula (I) wherein R1-R4 and p and q are as defined in the claims.

Cu(II)-mediated C-H amidation and amination of arenes: Exceptional compatibility with heterocycles

A Cu(OAc)2-mediated C-H amidation and amination of arenes and heteroarenes has been developed using a readily removable directing group. A wide range of sulfonamides, amides, and anilines function as amine donors in this reaction. Heterocycles present in both reactants are tolerated, making this a broadly applicable method for the synthesis of a family of inhibitors including 2-benzamidobenzoic acids and N-phenylaminobenzoates.

Synthesis and structure-activity relationships of o-sulfonamido- arylhydrazides as inhibitors of LL-diaminopimelate aminotransferase (LL-DAP-AT)

Recently, ll-diaminopimelate aminotransferase (ll-DAP-AT), a pyridoxal-5′-phosphate (PLP)-dependent enzyme, was reported to catalyze a key step in the biosynthesis of l-lysine in plants and Chlamydia. Previous screening of a 29201-compound library against