80704-02-5Relevant academic research and scientific papers
Palladium-catalyzed enantioselective C-H activation of aliphatic amines using chiral anionic BINOL-phosphoric acid ligands
Smalley, Adam P.,Cuthbertson, James D.,Gaunt, Matthew J.
supporting information, p. 1412 - 1415 (2017/02/10)
The design of an enantioselective Pd(II)-catalyzed C-H amination reaction is described. The use of a chiral BINOL phosphoric acid ligand enables the conversion of readily available amines into synthetically valuable aziridines in high enantiomeric ratios.
Pd-Catalyzed C-H aziridination of 3,3,5,5-tetrasubstituted piperazin-2-ones
Alanine, Thomas A.,Stokes, Stephen,Roberts, Craig A.,Scott, James. S.
, p. 53 - 56 (2017/12/27)
A palladium mediated C-H aziridination reaction of 3,3,5,5-substituted-piperazin-2-ones has been developed using phenyliodonium diacetate (PIDA) and succinic acid to give synthetically useful bicyclic aziridines, in moderate to good yields. Succinic acid
