808134-47-6Relevant articles and documents
Discovery of N1-(6-Chloroimidazo[2,1-b][1,3]-thiazole-5- sulfonyl)tryptamine as a potent, selective, and orally active 5-HT6 receptor agonist
Cole, Derek C.,Stock, Joseph R.,Lennox, William J.,Bernotas, Ronald C.,Ellingboe, John W.,Boikess, Steve,Coupet, Joseph,Smith, Deborah L.,Leung, Louis,Zhang, Guo-Ming,Feng, Xidong,Kelly, Michael F.,Galante, Rocco,Huang, Pingzhong,Dawson, Lee A.,Marquis, Karen,Rosenzweig-Lipson, Sharon,Beyer, Chad E.,Schechter, Lee E.
, p. 5535 - 5538 (2007)
N1-Arylsulfonyltryptamines have been identified as 5-HT 6 receptor ligands. In particular, N1(6-chloroimidazo[2,1- b][1,3]thiazole-5-sulfonyl)tryptamine (11q) is a high affinity, potent full agonist (5-HT6 Ksub
