817204-08-3Relevant articles and documents
Thio acid/azide amidation: An improved route to N-acyl sulfonamides
Barlett, Kristin N.,Kolakowski, Robert V.,Katukojvala, Sreenivas,Williams, Lawrence J.
, p. 823 - 826 (2007/10/03)
A one-pot procedure for the conversion of carboxylic acids to N-acyl sulfonamides, via thio acid/azide amidation, is presented. The method is compatible with acid- and base-sensitive amino acid protection. N-Acyl sulfonamide synthesis on solid support, pe