83195-24-8Relevant academic research and scientific papers
NOVEL DIPEPTIDYL-PEPTIDASE-IV INHIBITORS
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Paragraph 0072, (2013/07/25)
The invention comprises novel inhibitors of dipeptidyl peptidase IV (DPP-IV) with beta blocker activity, pharmaceutical compositions comprising therapeutically effective amounts of novel inhibitors of DPP-IV, and novel methods of treating medical conditio
COMPOUNDS AND METHOD FOR TREATMENT OR PROPHYLAXIS OF CARDIAC DISOREDRS
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, (2008/06/13)
A short-acting β-blocking compound of the formula STR1 wherein Ar may be substituted or unsubstituted aromatic, Y may be a straight or branched carbon chain or aralkyl, R may be lower alkyl, lower alkenyl, lower alkynyl, aryl or aralkyl, and x is an integer from 1 to about 3; or a pharmaceutically acceptable salt thereof.
Ultra-short-acting β-adrenergic receptor blocking agents. I. (Aryloxy)propanolamines containing esters in the nitrogen substituent
Erhardt,Woo,Gorczynski,Anderson
, p. 1402 - 1407 (2007/10/02)
In an attempt to produce short-acting β-adrenergic receptor blocking agents, we prepared several (aryloxy)propanolamines with ester functions incorporated into the nitrogen substituent. Many of these compounds exhibited a short duration of blocking activity after their continuous intravenous infusion for 40 min. However, their durations were found to increase considerably upon longer intravenous infusion.
