848469-63-6Relevant articles and documents
Synthesis and monoamine transporter affinity of new 2β-carbomethoxy- 3β-[4-(substituted thiophenyl)]phenyltropanes: Discovery of a selective SERT antagonist with picomolar potency
Tamagnan, Gilles,Alagille, David,Fu, Xing,Kula, Nora S.,Baldessarini, Ross J.,Innis, Robert B.,Baldwin, Ronald M.
, p. 1131 - 1133 (2007/10/03)
Preparation of cocaine analogues has been aimed largely at development of stable compounds with high affinity and selectivity for the dopamine transporter (DAT). We now report the synthesis and monoamine transporter affinity of 10 new 2β-carbomethoxy-3β-[