849343-65-3Relevant academic research and scientific papers
TRPV1 AGONISTS, FORMULATIONS CONTAINING THEM AND USES THEREOF
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Page/Page column 10-11, (2010/02/15)
The compounds of the general formula (I) in which X is represents two hydrogen atoms, a π-bond, oxygen or methylene; R2 is a C6-C12 aryl, or arylalkyl residue; R3 is hydrogen, 2-hydroxyethyl or 2-aminoethyl are useful for the treatme
Development of the first ultra-potent "capsaicinoid" agonist at transient receptor potential vanilloid type 1 (TRPV1) channels and its therapeutic potential
Appendino, Giovanni,De Petrocellis, Luciano,Trevisani, Marcello,Minassi, Alberto,Daddario, Nives,Moriello, Aniello Schiano,Gazzieri, David,Ligresti, Alessia,Campi, Barbara,Fontana, Gabriele,Pinna, Christian,Geppetti, Pierangeio,Di Marzo, Vincenzo
, p. 561 - 570 (2007/10/03)
Olvanil (N-9-Z-octadecenoyl-vanillamide) is an agonist of transient receptor potential vanilloid type 1 (TRPV1) channels that lack the pungency of capsaicin and was developed as an oral analgesic. Vanillamides are unmatched in terms of structural simplici
