86129-52-4Relevant articles and documents
Synthesis and structure-activity relationships of a series of benzazepine derivatives as 5-HT2C receptor agonists
Shimada, Itsuro,Maeno, Kyoichi,Kondoh, Yutaka,Kaku, Hidetaka,Sugasawa, Keizo,Kimura, Yasuharu,Hatanaka, Ken-ichi,Naitou, Yuki,Wanibuchi, Fumikazu,Sakamoto, Shuichi,Tsukamoto, Shin-ichi
, p. 3309 - 3320 (2008/09/20)
To identify potent and selective 5-HT2C receptor agonists, a series of novel benzazepine derivatives were synthesized, and their structure-activity relationships examined. The compounds were evaluated for their 5-HT2C, 5-HT2A/s