868372-53-6Relevant articles and documents
Discovery of pyrrolo[2,3-d]pyrimidin-4-ones as corticotropin-releasing factor 1 receptor antagonists with a carbonyl-based hydrogen bonding acceptor
Aso, Kazuyoshi,Kobayashi, Katsumi,Mochizuki, Michiyo,Kanzaki, Naoyuki,Sako, Yuu,Yano, Takahiko
, p. 2365 - 2371 (2011/05/15)
A new class of pyrrolo[2,3-d]pyrimidin-4-one corticotropin-releasing factor 1 (CRF1) receptor antagonists has been designed and synthesized. In general, reported CRF1 receptor antagonists possess a sp 2-nitrogen atom as hy