878384-17-9Relevant academic research and scientific papers
PROCESS FOR PREPARING SUBSTITUTED 1-O-ACYL-2-DEOXY-2-FLUORO-4-THIO-β-D-ARABINOFURANOSES
-
, (2011/07/07)
The present invention relates to a process for preparing 1-O-acyl-2-deoxy-2-fluoro-4-thio-??-D-arabinofuranoses having formula I and intermediates thereof: wherein R1 represents -C(O)-C1-C6-alkyl or -C(O)-aryl; and R2 represents C1-C6-alkyl, C1-C4-perfluo
PROCESS FOR PREPARING SUBSTITUTED 1-O-ACYL-2-DEOXY-2-FLUORO-4-THIO-BETA-D-ARABINOFURANOSES
-
, (2011/07/06)
The present invention relates to a process for preparing 1-O-acyl-2-deoxy-2-fluoro-4-thio-β-D-arabinofuranoses having formula I and intermediates thereof: wherein R1 represents —C(O)—C1-C6-alkyl or —C(O)-aryl; and R2
Process for preparing substituted 1-O-acyl-2-deoxy-2-fluoro-4-thio-?-D-arabinofuranoses
-
, (2011/12/03)
The present invention relates to a process for preparing 1-0-acyl-2-deoxy-2-fluoro-4-thio-β-D-arabinofuranoses in which R1 represents C(O)-C1-C6-alkyl or C(O)-aryl; R2 represents C1-C6-alkyl, C1-Csub
Synthesis and conformational analysis of 2′-fluoro-5-methyl-4′- thioarabinouridine (4′S-FMAU)
Watts, Jonathan K.,Sadalapure, Kashinath,Choubdar, Niloufar,Pinto, B. Mario,Damha, Masad J.
, p. 921 - 925 (2007/10/03)
An improved synthesis of 2′-deoxy-2′-fluoro-5-methyl-4′- thioarabinouridine (4′S-FMAU) is described. Participation of the 3′-O-benzoyl protecting group in the thiosugar precursor influenced the stereochemistry of the N-glycosylation reaction in nonpolar s
