887707-23-5Relevant articles and documents
AROMATIC RING DERIVATIVE AS IMMUNOREGULATION AND PREPARATION METHOD AND APPLICATION OF AROMATIC RING DERIVATIVE
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Paragraph 0299-0300, (2021/10/15)
Relating to a compound represented by formula (I) and a pharmaceutically acceptable salt of the compound, and an application of the compound as an S1P1 agonist.
Ligand-Promoted meta-C?H Functionalization of Benzylamines
Wang, Peng,Farmer, Marcus E.,Yu, Jin-Quan
supporting information, p. 5125 - 5129 (2017/04/24)
Meta-C?H functionalization of benzylamines has been developed using a PdII/transient mediator strategy. Using 2-pyridone ligands and 2-carbomethoxynorbornene (NBE-CO2Me) as the mediator, arylation, amination, and chlorination of benzylamines are realized. This protocol features a broad substrate scope and is compatible with heterocylic coupling partners. Moreover, the loading of the Pd can be lowered to 2.5 mol % by using the optimal ligand.
Substituted diazaspiroalkanes as androgen receptor modulators
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Page/Page column 19; 20; 21, (2016/08/10)
This invention provides for compounds of the Formula II: wherein A, B, Het, R1, R2 and R3 are as described herein. These compounds are androgen receptor modulators useful for the treatment of androgen receptor-associated conditions.