890831-59-1Relevant academic research and scientific papers
Synthesis and evaluation of a set of 4-Phenylpiperidines and 4-Phenylpiperazines as D2 receptor ligands and the discovery of the dopaminergic stabilizer 4-[3-(Methylsulfonyl)phenyl]-l-propylpiperidine (huntexil, pridopidine, ACR16)
Pettersson, Fredrik,Ponten, Henrik,Waters, Nicholas,Waters, Susanna,Sonesson, Clas
supporting information; experimental part, p. 2510 - 2520 (2010/08/22)
Modification of the partial dopamine type 2 receptor (D2) agonist 3-(l-benzylpiperidin-4-yl)phenol (9a) generated a series of novel functional D2 antagonists with fast-off kinetic properties. A representative of this series, pridopid
