903512-73-2Relevant academic research and scientific papers
Novel, orally bioavailable γ-aminoamide CC chemokine receptor 2 (CCR2) antagonists
Pasternak, Alexander,Marino, Dominick,Vicario, Pasquale P.,Ayala, Julia Marie,Cascierri, Margaret A.,Parsons, William,Mills, Sander G.,MacCoss, Malcolm,Yang, Lihu
, p. 4801 - 4804 (2007/10/03)
Through modification of a screening hit we have discovered a structurally distinct new lead, (2S)-N-[3,5-bis(trifluoromethyl)benzyl]-2-(4-fluorophenyl)-4- (4-phenylpiperidin-1-yl)butanamide (11), which has subsequently served as the departure point for an
