940950-95-8Relevant academic research and scientific papers
Synthesis of 2-oxazolines by in situ desilylation and cyclodehydration of β-hydroxyamides
Brandst?tter, Marco,Roth, Fabian,Luedtke, Nathan W.
, p. 40 - 51 (2016/09/09)
A powerful method for the synthesis of 2-oxazolines from silyl-protected β-hydroxyamides is reported. Using diethylaminosulfur trifluoride (DAST) or its tetrafluoroborate salt (XtalFluor-E), silyl-protected β-amidoalcohols can be in situ deprotected and d
Unified azoline and azole syntheses by optimized aza-wittig chemistry
Loos, Patrick,Ronco, Cyril,Riedrich, Matthias,Arndt, Hans-Dieter
supporting information, p. 3290 - 3315 (2013/06/27)
Intramolecular aza-Wittig ring closures were applied to synthesize thiazolines, oxazolines, and imidazolines from β-azido thioester, ester, and amide precursors. The cyclization precursors were obtained from amino acid derivatives. Optimized conditions fo
