945534-39-4Relevant academic research and scientific papers
New sst4/5-selective somatostatin peptidomimetics based on a constrained tryptophan scaffold
Feytens, Debby,Cescato, Renzo,Reubi, Jean Claude,Tourwé, Dirk
, p. 3397 - 3401 (2008/02/09)
The synthesis and biological evaluation of four peptidomimetic analogs of somatostatin based on a constrained Trp residue, 3-amino-indolo[2,3-c]azepin-2- one (Aia), are reported. It is shown that dipeptidomimetics with a D-Aia-Lys sequence, functionalized
