98976-81-9Relevant academic research and scientific papers
Directed Ortho Metalation of O-Pyridyl Carbamates. Regiospecific Entries into Polysubstituyed Pyridines
Miah, M. A. J.,Snieckus, V.
, p. 5436 - 5438 (1985)
Ortho-lithiated species of O-pyridyl carbamates 1a-c constitute new synthetic intermediates which provide a variety of polysubstituted pyridines (Table I) by reaction with electrophiles (2a-c) and anionic Fries rearrangement (3,4).Further metalation (7), ipso carbodestannylation (10, E=I, COMe), and reductive elimination of the carbamate directing group (56) are also described.
3-pyridyloxymethyl heterocyclic ether compounds useful in controlling neurotransmitter release
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, (2008/06/13)
Novel heterocyclic ether compounds of the formula: STR1 wherein n, *, R1, R2, R3 and y are specifically defined, or pharmaceutically acceptable salts or prodrugs thereof, which are useful in selectively controlling neurotransmitter release; therapeutically-effective pharmaceutical compositions of these compounds; and use of said compositions to selectively control neurotransmitter release in mammals.
