167298-58-0

Basic information

• Product Name: Cyclopentanol,3-amino-,(1R,3R)-rel-(9CI)
• Synonyms: Cyclopentanol,3-amino-,(1R,3R)-rel-(9CI);Trans-3-Aminocyclopentanol(WX600109)
• CAS NO: 167298-58-0
• Molecular Formula: C5H11NO
• Molecular Weight: 101.14694
• Product Categories: VARIOUSAMINE
• Mol File: 167298-58-0.mol

Chemical Properties

• Boiling Point: 179.4±33.0 °C(Predicted)
• Appearance: /
• Density: 1.084±0.06 g/cm3(Predicted)
• Storage Temp.: 2-8°C(protect from light)
• PKA: 15.06±0.40(Predicted)
• CAS DataBase Reference: Cyclopentanol,3-amino-,(1R,3R)-rel-(9CI)(CAS DataBase Reference)
• NIST Chemistry Reference: Cyclopentanol,3-amino-,(1R,3R)-rel-(9CI)(167298-58-0)
• EPA Substance Registry System: Cyclopentanol,3-amino-,(1R,3R)-rel-(9CI)(167298-58-0)

Safety Data

• Hazardous Substances Data: 167298-58-0(Hazardous Substances Data)

Usage

Uses

Used in Organic Chemistry:
Cyclopentanol,3-amino-,(1R,3R)-rel-(9CI) is used as a building block in the synthesis of various organic compounds. Its unique structure and stereochemistry allow for the creation of a wide range of molecules with diverse properties and applications.
Used in Pharmaceutical Research:
In the pharmaceutical industry, Cyclopentanol,3-amino-,(1R,3R)-rel-(9CI) is used as a starting material for the development of new drugs. Its specific stereochemistry plays a vital role in determining the compound's biological activity, making it a promising candidate for the design and synthesis of innovative pharmaceutical agents.
Used in Drug Synthesis:
Cyclopentanol,3-amino-,(1R,3R)-rel-(9CI) is utilized in the synthesis of drugs targeting specific medical conditions. Its unique structure and stereochemistry enable the development of drugs with improved efficacy, selectivity, and reduced side effects.
Used in Chiral Chemistry:
In the field of chiral chemistry, Cyclopentanol,3-amino-,(1R,3R)-rel-(9CI) is employed as a chiral building block for the synthesis of enantiomerically pure compounds. Its specific stereochemistry allows for the creation of chiral molecules with distinct biological activities and properties.
Used in Analytical Chemistry:
Cyclopentanol,3-amino-,(1R,3R)-rel-(9CI) can be used as a chiral reference standard in analytical chemistry. Its unique stereochemistry makes it a valuable tool for the identification and quantification of enantiomers in various samples.

Upstream product

• 1154870-59-3 (±)-trans-(3-hydroxycyclopentyl)carbamic acid tert-butyl ester 
• 939426-84-3 C₁₃H₁₇NO₃ 
• 160167-65-7 cis-3(S)-(N-D-Alanylamino)cyclopentan-1(R)-ol 
• 542-92-7 cyclopenta-1,3-diene 
• 126924-22-9 (1S,4R,αR-)-3-(α-hydroxyphenylacetyl)-2-oxa-3-aza-bicyclo[2,2,1]hept-5-ene 
• 207729-04-2 C₁₀H₁₉NO₃ 
• 207729-04-2 C₁₀H₁₉NO₃ 
• 121129-38-2 2-(tert-Butylglycoloyl)-3,6-dihydro-3,6-methano-2H-1,2-oxazine 
• 121129-35-9 2-Mandeloyl-3,6-dihydro-3,6-methano-2H-1,2-oxazine 

Downstream Products

• 1154870-59-3 trans-(+/-)-(3-hydroxycyclopentyl)-carbamic acid,1,1-dimethylethyl ester 
• 847416-99-3 tert-butyl N-(3-oxocyclopentyl)carbamate 
• 124555-33-5 (1S,3R)-3-aminocyclopentan-1-ol hydrochloride 
• 1610517-93-5 C₂₂H₂₅N₃O₅ 
• 1036260-18-0 (1S,3R)-3-aminocyclopentane-1-ol 
• 1110772-05-8 (1R,3S)-3-aminocyclopentan-1-ol 
• 167465-99-8 (1S,3R)-3-hydroxycyclopentyl-1-carbamic acid tert-butyl ester 
• 1279032-31-3 (1R,3S)-3-amino-1-cyclopentanol hydrochloride 

Relevant articles and documents

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The invention discloses a preparation method of (1R,3S)-3-aminocyclopentanol and an intermediate thereof. The invention provides a preparation method of a compound as shown in a formula I'-1. The preparation method comprises a step: re-crystallizing a mixture of compounds as shown in the formula I'-1 and the formula I'-2 in a solvent, wherein the solvent is a mixed solvent of a poor solvent and agood solvent, the poor solvent is a ketone solvent and methanol, and the good solvent is water. The preparation method is high in reaction yield, and a single-configuration product with high optical purity can be obtained.

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