trans-Hexahydroindolophenanthridines ("Benzergolines"), the First Structural Class of Potent and Selective Dopamine D1 Receptor Agonists Lacking a Catechol Group

Article abstract of DOI:10.1021/jm00105a047

In contrast to the many selective dopamine (DA) D₂ receptor agonists known, only two prototypes of selective D₁ receptor agonists have been described; both show preference for the periphery due to their catechol partial structures.Ou