Bioorganic and Medicinal Chemistry Letters p. 546 - 553 (2008)
Update date:2022-08-03
Topics:
Pfefferkorn, Jeffrey A.
Larsen, Scott D.
Huis, Chad Van
Sorenson, Roderick
Barton, Tom
Winters, Thomas
Auerbach, Bruce
Wu, Chenyan
Wolfram, Thaddeus J.
Cai, Hongliang
Welch, Kathleen
Esmaiel, Nadia
Davis, JoAnn
Bousley, Richard
Olsen, Karl
Mueller, Sandra Bak
Mertz, Thomas
Cholesterol absorption inhibition (CAI) represents an important treatment option for hypercholesterolemia. Herein, we report the design and evaluation of a series of substituted oxazolidinones as ligands for the Niemann Pick C1 Like 1 (NPC1L1) protein, a
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