Potent vasopressin antagonists lacking the proline residue at position 7

DOI: 10.1021/jm00156a015

Source and publish data:

Journal of Medicinal Chemistry p. 984 - 988 (1986)

Update date:2022-08-04

Topics:

Authors:

Ali Ali

Bryan Bryan

Chang Chang

Huffman Huffman

Moore Moore

Heckman Heckman

Kinter Kinter

McDonald

Schmidt Schmidt

Shue Shue

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Article abstract of DOI:10.1021/jm00156a015

As part of a program to design potent antidiuretic vasopressin antagonists and to define the minimum effective pharmacophore requirements for vasopressin (VP) antagonist activity, we studied the importance of the C-terminal tripeptide of a previously repo

Full text of DOI:10.1021/jm00156a015

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Product name:1,Val⁴,desPro⁷,desGly⁹>AVP

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