Potent vasopressin antagonists lacking the proline residue at position 7

DOI: 10.1021/jm00156a015

Source and publish data:

Journal of Medicinal Chemistry p. 984 - 988 (1986)

Update date:2022-08-04

Topics:

Authors:

Ali Ali

Bryan Bryan

Chang Chang

Huffman Huffman

Moore Moore

Heckman Heckman

Kinter Kinter

McDonald

Schmidt Schmidt

Shue Shue

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1021/jm00156a015

As part of a program to design potent antidiuretic vasopressin antagonists and to define the minimum effective pharmacophore requirements for vasopressin (VP) antagonist activity, we studied the importance of the C-terminal tripeptide of a previously repo

Full text of DOI:10.1021/jm00156a015

Products guided by the article

Product name:1,Val⁴,desPro⁷,desGly⁹>AVP

Cas No:101835-07-8

R&D Labs maybe for 101835-07-8

Tianjin Dongchang Fine Chemical Industry Co., Ltd.

Contact:+86-22-29894595

Address:Economic Developing Zone, Ji County, Tianjin, China
Shanghai shibo Chemical Co., Ltd

Contact:+86-021-60753516

Address:688 Qiushi Road, Jinshan High-tech Park, Shanghai, China,201512
Jiangsu Jiuri Chemical Co.,Ltd.

Contact:+86-519-82118868

Address:Tianwang Town, Jurong City, Jiangsu Province, China
Onlychem (Jinan)Biotech Co.,Ltd

Contact:86-531-83175885

Address:No. 44, Honglou South Road, Jinan,China
Shanghai Hanshare Industry Co.,Ltd.

Contact:86 21 20960688

Address:RM902-903,Building E, Wanda Plaza,No.26,Zhoukang Road, Pudong District, Shanghai, China

Relevant to this article

Doi:10.1039/jr9570001998
()
Discovery of a Potent, Selective Renal Sodium-Dependent Glucose Cotransporter 2 (SGLT2) Inhibitor (HSK0935) for the Treatment of Type 2 Diabetes

Doi:10.1021/acs.jmedchem.6b01818
(2017)
Total synthesis of ouabagenin and ouabain

Doi:10.1002/anie.200704959
(2008)
Ligand-Controlled Regiodivergent Hydroformylation of Ynamides: A Stereospecific and Regioselective Access to 2- And 3-Aminoacroleins

Doi:10.1021/acs.orglett.9b03566
(2019)
Discovery of novel dual inhibitors of the wild-type and the most prevalent drug-resistant mutant, S31N, of the M2 proton channel from influenza A virus

Doi:10.1021/jm301538e
(2013)
94. Synthesen von Dibenzo<1,4>dioxin-2,3-chinonen, einschliesslich der Ecklonochinone A und B sowie der Isoecklonochinone A und B

Doi:10.1002/hlca.19850680407
(1985)

Article Doi