BENZOXADIAZOCINES, BENZOTHIADIAZOCINES AND BENZOTRIAZOCINES-V; THE SYNTHESIS OF SOME 2-AMINO-6-METHYL- AND 2-AMINO-6-PHENYL-5,6-DIHYDRO-4H-3,1,6-BENZOTHIADIAZOCINES

Article abstract of DOI:10.1016/S0040-4020(01)96604-9

A method is described for the synthesis of hydrochlorides of some type 8 title compounds in which the nucleophilicity of N-2 is reduced or completely lost so as to prevent ring contraction reactions and, as a result, making these compounds comparatively s