Organic Letters p. 4156 - 4159 (2010)
Update date:2022-07-30
Topics:
Zhu, Qiang
Lu, Yixin
A facile synthesis of chiral bicyclic amidines and imidazolines from readily available 1,2-diamines has been developed. The reported synthetic strategy relies on an intramolecular cyclization which involves a carboxylic amide derived imidoyl chloride as a
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