Bioorganic and Medicinal Chemistry Letters p. 869 - 873 (2011)
Update date:2022-07-30
Topics:
Tyagarajan, Sriram
Chakravarty, Prasun K.
Park, Min
Zhou, Bishan
Herrington, James B.
Ratliff, Kevin
Bugianesi, Randall M.
Williams, Brande
Haedo, Rodolfo J.
Swensen, Andrew M.
Warren, Vivien A.
Smith, McHardy
Garcia, Maria
Kaczorowski, Gregory J.
McManus, Owen B.
Lyons, Kathryn A.
Li, Xiaohua
Madeira, Maria
Karanam, Bindhu
Green, Mitchell
Forrest, Michael J.
Abbadie, Catherine
McGowan, Erin
Mistry, Shruti
Jochnowitz, Nina
Duffy, Joseph L.
N-type calcium channels (Cav2.2) have been shown to play a critical role in pain. A series of low molecular weight 2-aryl indoles were identified as potent Cav2.2 blockers with good in vitro and in vivo potency.
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