Antiandrogenic steroidal sulfonylpyrazoles

DOI: 10.1021/jm00170a008

Source and publish data:

Journal of Medicinal Chemistry p. 2094 - 2100 (1990)

Update date:2022-08-04

Topics:

Authors:

Christiansen

Bell Bell

D'Ambra D'Ambra

Mallamo Mallamo

Herrmann

Ackerman

Opalka Opalka

Kullnig Kullnig

Winneker

Snyder Snyder

Batzold Batzold

Schane Schane

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1021/jm00170a008

The steroidal sulfonylpyrazole 1 bound to the rat ventral prostate androgen receptor in vitro; it inhibited testosterone propionate induced increases in ventral prostate weight in vivo in the castrated, immature male rat with an ED₅₀ of 15 mg/k

Full text of DOI:10.1021/jm00170a008

Products guided by the article

Product name:(1R,3aS,3bR,5aS,10aS,10bS,12aS)-1-Ethynyl-7-methanesulfonyl-10a,12a-dimethyl-1,2,3,3a,3b,4,5,5a,6,7,10,10a,10b,11,12,12a-hexadecahydro-7,8-diaza-dicyclopenta[a,h]phenanthren-1-ol

Cas No:127881-88-3

R&D Labs maybe for 127881-88-3

Hangzhou Pharma & Chem Co.,Ltd.

Contact:+86-571-87040515

Address:No,139Qingchun Rd
Chinapeptides Co,. Ltd

Contact:+86-021-50792271

Address:Building 24A, 300 Chuantu Road, Chuansha, Pudong new area, Shanghai, China, 201202
Shanghai FWD Chemicals ltd

website:http://www.fwdchem.com

Contact:86-21-54450828

Address:Room 802,Lotus Tower ,159 Tianzhou Road,Xuhui District,Shanghai
Nantong Chem-land Co., Ltd.

Contact:86 513 85512619

Address:Rm.1306, Building A, Wenfeng Mansion,168 Gongnong Road, Nantong Jiangsu China
Xian Changyue Biological Technology Co., Ltd.

website:https://www.xachangyue.com/

Contact:+86-029-88211911

Address:Keji Road NO.70

Relevant to this article

STRUCTURE OF FR 900483, A NEW IMMUNOMODULATOR ISOLATED FROM A FUNGUS

Doi:10.1016/S0040-4039(00)82028-6
(1988)
Di(methylimidazole)prolinol silyl ether catalyzed highly Michael addition of aldehydes to nitroolefins in water

Doi:10.1021/ol901204b
(2009)
Iridium-catalyzed isomerization of primary allylic alcohols under mild reaction conditions

Doi:10.1016/j.tetlet.2009.04.130
(2009)
Diverting β-Hydride Elimination of a ?-Allyl Pd^IICarbene Complex for the Assembly of Disubstituted Indolines via a Highly Diastereoselective (4 + 1)-Cycloaddition

Doi:10.1021/acs.orglett.0c02374
(2020)
Stereoselective synthesis of N-heterocycles: application of the asymmetric Cu-catalyzed addition of Et₂Zn to functionalized alkyl and aryl imines

Doi:10.1016/j.tet.2009.04.002
(2009)
Total synthesis and absolute configuration of the natural amino acid tetrahydrolathyrine

Doi:10.1021/jo900800x
(2009)

Article Doi