Specific Bradycardic Agents. 2. Heteroaromatic Modifications in the Side Chain of Specific Bradycardic Benzazepinones: Chemistry, Pharmacology, and Structure-Activity Relationships

DOI: 10.1021/jm00107a011

Source and publish data:

Journal of Medicinal Chemistry p. 942 - 947 (1991)

Update date:2022-08-02

Topics:

Authors:

Bomhard, Andreas

Reiffen, Manfred

Heider, Joachim

Psiorz, Manfred

Lillie, Christian

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Article abstract of DOI:10.1021/jm00107a011

Compound 1 (UL-FS 49) has recently been described as the representative of a novel class of antiischemic compounds termed "specific bradycardic agents".In search of specific bradycardic agents with different pharmacokinetic profiles, heteroaromatic analog

Full text of DOI:10.1021/jm00107a011

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