7-Azetidinylquinolones as antibacterial agents. Synthesis and structure- activity relationships

DOI: 10.1021/jm00059a002

Source and publish data:

Journal of Medicinal Chemistry p. 801 - 810 (1993)

Update date:2022-08-03

Topics:

Authors:

Frigola Frigola

Pares Pares

Corbera Corbera

Vano Vano

Merce Merce

Torrens Torrens

Mas Mas

Valenti Valenti

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Article abstract of DOI:10.1021/jm00059a002

A series of novel antibacterial quinolones and naphthyridones has been prepared which contain 7-azetidinyl substituents in place of the usual piperazine or aminopyrrolidine groups. These azetidinyl derivatives were evaluated for in vitro activity by deter

Full text of DOI:10.1021/jm00059a002

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