
Tetrahedron Letters p. 5263 - 5264 (1991)
Update date:2022-08-04
Topics:
Rivero
Greenlee
Patchett
As part of an effort to design human renin inhibitors with improved bioavailability, the amino-terminal Phe-His element present in many classes of renin inhibitors was replaced by a sulfone containing isostere.
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