Synthesis and biological activity of new 2,3-dihydro-1H-cyclopenta[b]- quinoline derivatives as acetylcholinesterase inhibitors

DOI: 10.2174/157018012801319454

Source and publish data:

Letters in drug design and discovery p. 645 - 654 (2012)

Update date:2022-08-04

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Authors:

Szymanski, Pawel

Markowicz, Magdalena

Bajda, Marek

Malawska, Barbara

Mikiciuk-Olasik, Elzbieta

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Article abstract of DOI:10.2174/157018012801319454

In this study we present synthesis and biological evaluation of derivatives of 4-fluorobenzoic acid and 2,3-dihydro-1H-cyclopenta[b]quinoline towards inhibition of acetylcholinesterase (AChE) and butyrylcholinesterase (BChE). Synthesis of acquired molecul

Full text of DOI:10.2174/157018012801319454

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