Ring opening of cyclic sulfamidates with magnesiated heterocycles: Expedient synthesis of highly functionalised azaindolines and azatetrahydroquinolines

DOI: 10.1055/S-0032-1317170

Source and publish data:

Synlett p. 2408 - 2412 (2012)

Update date:2022-08-05

Topics:

Authors:

Moss, Thomas A.

Hayter, Barry R.

Hollingsworth, Ian A.

Nowak, Thorsten

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Article abstract of DOI:10.1055/S-0032-1317170

Magnesiated chloropyrimidine and chloropyridine derivatives, obtained by deprotonation with TMPMgCl·LiCl at room temperature, undergo facile ring-opening reactions with five- and six-membered N-Boc and N-Bn cyclic sulfamidates. After an acidic workup, the

Full text of DOI:10.1055/S-0032-1317170

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