Pyrrolo[2,1-c][1,4]benzodiazepines: A mild conversion of thiolactam into amidine

DOI: 10.1016/S0040-4039(00)78862-9

Source and publish data:

Tetrahedron Letters p. 2803 - 2804 (1992)

Update date:2022-08-03

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Authors:

Foloppe, Mari P.

Rault, Sylvain

Robba, Max

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Article abstract of DOI:10.1016/S0040-4039(00)78862-9

Reaction of 2-hydoxy pyrrolo [2,1-c] [1,4] benzodiazepines-5-one-thione or 5,11-dithiones with ammonia in presence of mercuric chloride affords new amidines in high yield.

Full text of DOI:10.1016/S0040-4039(00)78862-9

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