Pyrrolo[2,1-c][1,4]benzodiazepines: A mild conversion of thiolactam into amidine

DOI: 10.1016/S0040-4039(00)78862-9

Source and publish data:

Tetrahedron Letters p. 2803 - 2804 (1992)

Update date:2022-08-03

Topics:

Authors:

Foloppe, Mari P.

Rault, Sylvain

Robba, Max

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/S0040-4039(00)78862-9

Reaction of 2-hydoxy pyrrolo [2,1-c] [1,4] benzodiazepines-5-one-thione or 5,11-dithiones with ammonia in presence of mercuric chloride affords new amidines in high yield.

Full text of DOI:10.1016/S0040-4039(00)78862-9

Products guided by the article

Product name:Benzoic acid (R)-5,11-dioxo-2,3,5,10,11,11a-hexahydro-1H-benzo[e]pyrrolo[1,2-a][1,4]diazepin-2-yl ester

Cas No:142558-31-4

R&D Labs maybe for 142558-31-4

Exploiter Molybdenum Co.,Ltd

Contact:86-379-63338609

Address:Jiudian Village,Deting Town,Song County,Luoyang
Jiangxi Dongxu Chemical Science & Technology Co.,Ltd

Contact:+86-791-86899381

Address:Nanchang, Jiangxi, China
Cangzhou Senary Chemical Science-tech Co., Ltd

Contact:+86-317-3563899, 3563699

Address:168 Jinde Road, Cangzhou, Hebei, China
TAIXING BEST NEW MATERIALS CO., LTD

Contact:0523-87998158;

Address:No.18 Zhonggang Road，Taixing City ，Jiangsu , China
Nanjing Legend Pharmaceutical & Chemical Co., Ltd.

Contact:+86-25-83767696

Address:14-7 Zhongshan Lu Guluo District, Nanjing

Relevant to this article

Pd-catalyzed tandem sp²-sp³ coupling reactions of chiral stannolanes: An efficient preparation of optically active tetrahydrobenz[f]isoindoles

Doi:10.1021/ol4003948
(2013)
Antioxidant activities of thiosemicarbazones from substituted benzaldehydes and N-(tetra-O-acetyl-β-d-galactopyranosyl)thiosemicarbazide

Doi:10.1016/j.ejmech.2012.10.004
(2013)
A flexible and modular stereoselective synthesis of (9R,10S)- dihydrosterculic acid

Doi:10.1016/j.tetasy.2013.01.003
(2013)
Practical Preparation of Chiral 4-Substituted 2-Oxazolidinones

Doi:10.1246/cl.1992.991
(1992)
Discovery of a novel series of quinolone α7 nicotinic acetylcholine receptor agonists

Doi:10.1016/j.bmcl.2013.01.070
(2013)
Synthesis of new derivatives of pyrimido[5,4-e][1,2,4]triazolo[3,4-b] [1,3,4]thiadiazine and their enzyme inhibitory activity assessment on soybean 15-lipoxygenase

Doi:10.3184/174751912X13549029453945
(2013)

Article Doi