Pyrrolo[2,1-c][1,4]benzodiazepines: A mild conversion of thiolactam into amidine

DOI: 10.1016/S0040-4039(00)78862-9

Source and publish data:

Tetrahedron Letters p. 2803 - 2804 (1992)

Update date:2022-08-03

Topics:

Authors:

Foloppe, Mari P.

Rault, Sylvain

Robba, Max

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/S0040-4039(00)78862-9

Reaction of 2-hydoxy pyrrolo [2,1-c] [1,4] benzodiazepines-5-one-thione or 5,11-dithiones with ammonia in presence of mercuric chloride affords new amidines in high yield.

Full text of DOI:10.1016/S0040-4039(00)78862-9

Products guided by the article

Product name:Benzoic acid (R)-5,11-dioxo-2,3,5,10,11,11a-hexahydro-1H-benzo[e]pyrrolo[1,2-a][1,4]diazepin-2-yl ester

Cas No:142558-31-4

R&D Labs maybe for 142558-31-4

He Bei Shun Er Chemical Co., LTD.

Contact:86-0311-86996932/86860168

Address:No 18,North street
Synchem Pharma Co.,Ltd(expird)

Contact:+0086-21-61984905-1

Address:Building 60,Zimian Park, LongYang industrial Area, 1515Nong，Yuandong Road Fengxian District, Shanghai ,China
Tomo Pharma Chem Co., Limited

Contact:+86-158-05817090

Address:ROOM 9F, FLAT 2, GUODU DEVELOPING BLDG, No.182, ZHAOHUI ROAD
Greenutra Resource Inc

website:http://www.greenutra.cn

Contact:0086-411-39553357

Address:No. 7-1-1802, Huizhi Garden,Ocean Square,Dalian, 116033, China
XI'AN CHUKANG BIOTECHNOLOGY CO.,LTD

Contact:29-63685658 63685359

Address:Room 3-1202,Building 1,Oriental oasis,East of Xianning Road,Xi'an,Shaanxi 710043 P.R.China

Relevant to this article

Pd-catalyzed tandem sp²-sp³ coupling reactions of chiral stannolanes: An efficient preparation of optically active tetrahydrobenz[f]isoindoles

Doi:10.1021/ol4003948
(2013)
Antioxidant activities of thiosemicarbazones from substituted benzaldehydes and N-(tetra-O-acetyl-β-d-galactopyranosyl)thiosemicarbazide

Doi:10.1016/j.ejmech.2012.10.004
(2013)
A flexible and modular stereoselective synthesis of (9R,10S)- dihydrosterculic acid

Doi:10.1016/j.tetasy.2013.01.003
(2013)
Practical Preparation of Chiral 4-Substituted 2-Oxazolidinones

Doi:10.1246/cl.1992.991
(1992)
Discovery of a novel series of quinolone α7 nicotinic acetylcholine receptor agonists

Doi:10.1016/j.bmcl.2013.01.070
(2013)
Synthesis of new derivatives of pyrimido[5,4-e][1,2,4]triazolo[3,4-b] [1,3,4]thiadiazine and their enzyme inhibitory activity assessment on soybean 15-lipoxygenase

Doi:10.3184/174751912X13549029453945
(2013)

Article Doi