6-Alkyl-12-formylindolo[2,1-a]isoquinolines. Syntheses, estrogen receptor binding affinities, and stereospecific cytostatic activity

DOI: 10.1021/jm00097a011

Source and publish data:

Journal of Medicinal Chemistry p. 3537 - 3547 (1992)

Update date:2022-08-05

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Authors:

Polossek

Ambros Ambros

Von Angerer

Brandl Brandl

Mannschreck

Von Angerer

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Article abstract of DOI:10.1021/jm00097a011

A number of 6-alkyl-12-formyl-5,6-dihydroindolo[2,1-a]isoquinolines were synthesized by the Bischler-Napieralski reaction from the respective 1-alkyl- 2-(3-methoxyphenyl)ethylamines and bromo-substituted (methoxyphenyl)acetic acid chlorides followed by a

Full text of DOI:10.1021/jm00097a011

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