1-Substituted 2-benzylaminobenzimidazole derivatives: Compounds with H1-antihistamine activity

DOI: 10.1016/0223-5234(92)90153-R

Source and publish data:

European Journal of Medicinal Chemistry p. 395 - 400 (1992)

Update date:2022-07-31

Topics:

Authors:

Da Settimo

Primofiore

Da Settimo

Calzolari

Cazzulani

Passoni Passoni

Tofanetti

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Article abstract of DOI:10.1016/0223-5234(92)90153-R

The preparation of 1-substituted 2-benzylaminobenzimidazole derivatives 13-24 is described. Although these compounds have a different structure from the general structure I of antihistamines, they showed some antihistaminic activity (pA₂: 5-7)

Full text of DOI:10.1016/0223-5234(92)90153-R

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