Development of a Model for the δ Opioid Receptor Pharmacophore. 1. Conformationally Restricted Tyr1 Replacements in the Cyclic δ Receptor Selective Tetrapeptide Tyr-cOH (JOM-13)

DOI: 10.1021/jm00051a015

Source and publish data:

Journal of Medicinal Chemistry p. 4371 - 4383 (1994)

Update date:2022-08-04

Topics:

Authors:

Mosberg, Henry I.

Lomize, Andrei L.

Wang, Chenguang

Kroona, Heather

Heyl, Deborah L.

et al. et al.

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Article abstract of DOI:10.1021/jm00051a015

A series of analogues of the conformationally restricted δ opioid receptor selective tetrapeptide Tyr-cOH (JOM 13) was prepared in which the conformationally labile Tyr residue was replaced with several less flexible tyrosine analogues.Am

Full text of DOI:10.1021/jm00051a015

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