Development of a Model for the δ Opioid Receptor Pharmacophore. 1. Conformationally Restricted Tyr1 Replacements in the Cyclic δ Receptor Selective Tetrapeptide Tyr-cOH (JOM-13)

DOI: 10.1021/jm00051a015

Source and publish data:

Journal of Medicinal Chemistry p. 4371 - 4383 (1994)

Update date:2022-08-04

Topics:

Authors:

Mosberg, Henry I.

Lomize, Andrei L.

Wang, Chenguang

Kroona, Heather

Heyl, Deborah L.

et al. et al.

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1021/jm00051a015

A series of analogues of the conformationally restricted δ opioid receptor selective tetrapeptide Tyr-cOH (JOM 13) was prepared in which the conformationally labile Tyr residue was replaced with several less flexible tyrosine analogues.Am

Full text of DOI:10.1021/jm00051a015

Products guided by the article

Product name:1-Acetyl-5-hydroxy-3-(4-methoxy-phenyl)-pyrrolidine-2,2-dicarboxylic acid diethyl ester

Cas No:159391-37-4

R&D Labs maybe for 159391-37-4

HANGZHOU ZHONGCHANG SCIENTIFIC CO.,LTD

Contact:+86-571-88932183

Address:Hangzhou
ZUNYI CITY BEI YUAN CHEMICAL CO., LTD

website:http://www.china-beiyuan.com

Contact:+86-851-27751258

Address:Shawan Town, Huichuan District, Zunyi City, Guizhou Province, China
shanghai payne pharm co.,ltd.

Contact:+86-021-58123769

Address:No.780 of Cailun Road,Zhangjiang Hi-tech Park,Pudong,Shanghai
Anhui Charm Imp.&Exp.Co., Ltd

website:http://www.chinacharm.cn/

Contact:86 551 5316260

Address:No. 211,XiangZhang Road,Hefei City,Anhui Province,China
WUHAN WELLSONG INT'L CO.,LTD

Contact:+86-27-85733560

Address:NO.308,QINGNIAN RD.,WUHAN,CHINA

Relevant to this article

Spin Transition in [Fe(DPEA)(NCS)₂], a Compound with the New Tetradentate Ligand (2-Aminoethyl)bis(2-pyridylmethyl)amine (DPEA): Crystal Structure, Magnetic Properties, and M?ssbauer Spectroscopy

Doi:10.1021/ic9615133
(1997)
Doi:10.1021/jo01256a028
(1969)
A new synthetic route to 2-substituted naphtho[2,3-b]furan-4,9-dione

Doi:10.1002/jhet.5570340209
(1997)
Imidazo-oxazaphosphorines as precursors to chiral phosphite triesters

Doi:10.1080/07328319808003465
(1998)
Spectroscopic and crystallographic studies of phosphino adducts of gallium(III) iodide

Doi:10.1139/v97-038
(1997)
Synthesis and reactivity of 7,9-diphenyl-nido-carbaundecaboranes: Rearrangement processes in carbaplatinaboranes revisited

Doi:10.1039/a607523a
(1997)

Article Doi