CCK-A Receptor Selective Antagonists Derived from the CCK-A Receptor Selective Tetrapeptide Agonist Boc-Trp-Lys(Tac)-Asp-MePhe-NH2 (A-71623)

DOI: 10.1021/jm00001a027

Source and publish data:

Journal of Medicinal Chemistry p. 207 - 211 (1995)

Update date:2022-08-03

Topics:

Authors:

Sugg, Elizabeth E.

Kimery, Millard J.

Ding, Jian Mei

Kenakin, Deborah C.

Miller, Laurence J.

et al. et al.

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Article abstract of DOI:10.1021/jm00001a027

Analogs of the CCK-A receptor selective agonist Boc-Trp-Lys(Tac)-Asp-MePhe-NH2 (A-71623) were prepared in which the lysine residue was replaced with L-4-aminophenylalanine and D- or L-3-aminophenylalanine.These new analogs were moderately potent antagonis

Full text of DOI:10.1021/jm00001a027

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Product name:H-Trp-L-3-Amf<(N^ε-o-tolylamino)carbonyl>-Asp-MePh-NH2

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