Synthesis of substance-P C-terminal hexapeptide analogues and their biological activity. Analogues with antagonistic activity without containing D-amino acids

DOI: 10.1016/0223-5234(94)90028-0

Source and publish data:

European Journal of Medicinal Chemistry p. 667 - 673 (1994)

Update date:2022-08-05

Topics:

Authors:

Karagiannis

Manopoulou

Poulos Poulos

Stavropoulos

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Article abstract of DOI:10.1016/0223-5234(94)90028-0

Analogues of the C-terminal hexapeptide of substance P have been synthesized in which each amino-acid residue was replaced by the bulky and strong lipophilic residue Asp(OBzl). The amino-acid residue of other selected places has also been replaced by Glu(

Full text of DOI:10.1016/0223-5234(94)90028-0

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