Asymmetric Synthesis of cis -(S, R)-3-Amino-4-fluoro-1-methylpyrrolidine

DOI: 10.1055/s-0037-1611553

Source and publish data:

Synlett p. 1228 - 1230 (2019)

Update date:2022-07-31

Topics:

Authors:

Bian, Jianwei

Cheung, Chiming

Fei, Zhongbo

Gao, Hongjun

Liu, Weipeng

Shen, Qirong

Xiong, Xin

Zhang, Jinzhu

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Article abstract of DOI:10.1055/s-0037-1611553

The development of the stereoselective synthesis of cis -(S, R)-3-amino-4-fluoro-1-methylpyrrolidine is described starting from chiral, non-racemic 1-[(3 S,4 S)-3-azido-4-hydroxypyrrolidin-1-yl]-2,2,2-trifluoroethan-1-one. Two sets of deoxyfluorination co

Full text of DOI:10.1055/s-0037-1611553

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Product name:6-Oxa-3-azabicyclo[3.1.0]hexane, 3-(trifluoroacetyl)- (9CI)

Cas No:164931-85-5

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