Resolution, EPC-Syntheses, Absolute Stereochemistry, and Pharmacology of the (S)-(+)- and (R)-(-)-Isomers of the MAO-A Inhibitor Tetrindole Hydrochloride

DOI: 10.1002/ardp.19953280710

Source and publish data:

Archiv der Pharmazie p. 619 - 622 (1995)

Update date:2022-08-04

Topics:

Authors:

Boes, Michael

Canesso, Rolf

Kettler, Rolf

Keller, Hans H.

Schoenholzer, Peter

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1002/ardp.19953280710

Resolution of (RS)-tetrindole (3) and enantioselective reductions of the imine 7 yielded (S)-(+)-(4) and (R)-(-)-tetrindole (5).The absolute stereochemistry of 4 was established by X-ray analysis of the corresponding Mosher amide 6.From in vitro as well a

Full text of DOI:10.1002/ardp.19953280710

Products guided by the article

Product name:8-Cyclohexyl-2,4,5,6-tetrahydro-1H-pyrazino<3,2,1-jk>carbazole

Cas No:171112-90-6

R&D Labs maybe for 171112-90-6

JIANGXI AIFEIMU TECHNOLOGY CO.，LTD

Contact:+86-570-6040289

Address:FINECHEMICAL PARK,ZIBU TOWN,WANNIAN COUNTY,JIANGXI PROV.,CHINA,ZIP
Shandong Wanda Organosilicon New Material Co., Ltd

Contact:+86-21-54177116;54302881

Address:R1318 Greenland No. 3 Lane 58 Xinjian East Rd., Minhang
Shanghai Pengkai Chemical Co.,Ltd

Contact:+86-21-60526671

Address:No.4226 Duzhuang Rd Minhang District Shanghai China
Nanjing Raise Pharmatech Co., Ltd

website:http://www.raisechem.com

Contact:+86-25-58649566

Address:B381,No.606,Ningliu Road,Jiangbei New Area,Nanjing,Jiangsu Province,China
Guangzhou Chemical Reagent Factory

Contact:+86-20-8435 9820 or 8435 7345

Address:Southern Guangzhou, Guangdong, China

Relevant to this article

Potential anti-inflammatory actions of the elmiric (lipoamino) acids

Doi:10.1016/j.bmc.2007.03.026
(2007)
2,3-Disubstituted indoles from olefins and hydrazines via tandem hydroformylation-Fischer indole synthesis and skeletal rearrangement

Doi:10.1039/b513364e
(2006)
(Hydroxyphenyl)oxazoline: A novel and remarkably facile entry into the area of chiral cationic alkylzirconium complexes which serve as polymerization catalysts

Doi:10.1021/om00011a010
(1995)
Unexpected reactions of anionic intermediates [(μ-RE)(μ-S=CS)Fe₂(CO)₆]^- with so₂Cl₂. Synthesis and characterization of novel dithioformato-bridged double clusters [(μ-RE)Fe₂(CO)₆]₂(μ-S=CS-μ) (E = S, Se)

Doi:10.1021/om960775+
(1997)
Doi:10.1002/hlca.19590420732
(1959)
A convenient synthesis of 2-alkyl-3-aryl-2,3-dihydro-1H-isoindol-1-ones by the reaction of N-alkyl-N-[(2-bromophenyl)methyl]benzamides with butyllithium

Doi:10.1016/j.tet.2016.06.082
(2016)

Article Doi