An easy entry to (1S, 2S) and (1R, 2R)-threo-Ifenprodil

Article abstract of DOI:10.1080/00397910008087268

A facile and practical synthesis of enantiomerically pure (L) or (D)-threo-Ifenprodil was accomplished from (1S, 2S)- and (1R, 2R)-threo-1-(p-nitrophenyl)-2-amino-propan-1, 3-diol via 3-phenylthio derivatives followed by Raney nickel reduction and convers

Full text of DOI:10.1080/00397910008087268

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Synthetic Communications: An
International Journal for Rapid
Communication of Synthetic
Organic Chemistry
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An Easy Entry to (1S, 2S) and
(1R, 2R)-Threo-Ifenprodil
Sergio Mantegani a , Emanuele Arlandini a , Enzo
Brambilla a , Paolo Cremonesi a & Mario Varasi a
a Pharmacia & Upjohn Department of Chemistry,
Discovery Research Oncology Viale Pasteur,
10-20014, Nerviano, MI, Italy
Published online: 04 Dec 2007.
To cite this article: Sergio Mantegani , Emanuele Arlandini , Enzo Brambilla ,
Paolo Cremonesi & Mario Varasi (2000) An Easy Entry to (1S, 2S) and (1R, 2R)-
Threo-Ifenprodil, Synthetic Communications: An International Journal for
Rapid Communication of Synthetic Organic Chemistry, 30:19, 3543-3553, DOI:
10.1080/00397910008087268
To link to this article: http://dx.doi.org/10.1080/00397910008087268
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